Comment · Sat, January 3, 2015 · Ceretropic
how would you classify tianeptine as?
Original post in this thread
nutrop · 2 points
Since it is uncontrolled in the U.S., it is being sold as a nootropic, but it sometimes fall under as TCA (tricyclic antidepressant) and as analgesic affecting the opioid receptor.
What they were answering
DrMichaelPLudwig · 1 points
The only literature currently touching its binging affininities is the original article that discovered discovered the affinities that lead to the current mu and deltal Ki values that we have.
In my own research, tianeptine completely substituted for butryfententanyl and acetylfentanyl in mice. A weak opioid would not do that. Also through speaking with a colleague, confidentially, who has an opioid problem, I was informed that .1g of tianeptine injected intravenously is almost indistinguishable from .1g of heroin injected intravenously. He said the charecteristic "rush" and "nod" are exactly the same. It's sad actually, he uses tianeptine, as well as other synth opioids to avoid giving a positive drug test and thus losing his job and professional license, but the tianeptine has done more venous damage in a few months than heroin did over years of use.
u/MisterYouAreSoDumb · Ceretropic
In my own research, tianeptine completely substituted for butryfententanyl and acetylfentanyl in mice.
You have to be trolling us now! Tianeptine substitutes for acetylfentanyl?!? The oral analog of the substance responsible for countless overdoses, because it was cut in Heroin, and people did not know it? The substance that is 15 times more potent than heroin?!? Fucking Tianeptine completely substitutes for acetylfentanyl? What was your study design for this mouse test?